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MedKoo Cat#: 576350 | Name: Tiamenidine hydrochloride

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tiamenidine hydrochloride is a centrally-acting alpha1 adrenergic receptor antagonist.

Chemical Structure

Tiamenidine hydrochloride
Tiamenidine hydrochloride
CAS#51274-83-0

Theoretical Analysis

MedKoo Cat#: 576350

Name: Tiamenidine hydrochloride

CAS#: 51274-83-0

Chemical Formula: C8H11Cl2N3S

Exact Mass: 251.0051

Molecular Weight: 252.16

Elemental Analysis: C, 38.11; H, 4.40; Cl, 28.12; N, 16.66; S, 12.71

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
HOE 42-440; HOE440; HOE-440; HOE 440; Sundralen; Symcor; Tiamenidine hydrochloride; Tiamenidine HCl; Thiamenidine hydrochloride; Thiamenidine HCl
IUPAC/Chemical Name
2-Imidazoline, 2-((2-chloro-4-methyl-3-thienyl)amino)-, monohydrochloride
InChi Key
RPZYVGSSBVNVCS-UHFFFAOYSA-N
InChi Code
InChI=1S/C8H10ClN3S.ClH/c1-5-4-13-7(9)6(5)12-8-10-2-3-11-8;/h4H,2-3H2,1H3,(H2,10,11,12);1H
SMILES Code
Cl.Cc1csc(Cl)c1NC2=NCCN2
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 252.16 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Kobinger W. Rudolf Buchheim lecture. Drugs as tools in research on adrenoceptors. Naunyn Schmiedebergs Arch Pharmacol. 1986 Feb;332(2):113-23. Review. PubMed PMID: 3010138. 2: Struthers AD, Dollery CT. Central nervous system mechanisms in blood pressure control. Eur J Clin Pharmacol. 1985;28 Suppl:3-11. Review. PubMed PMID: 2865146. 3: Reid JL, Campbell BC, Hamilton CA. Withdrawal reactions following cessation of central alpha-adrenergic receptor agonists. Hypertension. 1984 Sep-Oct;6(5 Pt 2):II71-5. Review. PubMed PMID: 6150002.

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