MedKoo Cat#: 412893 | Name: Cilobamine mesylate

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Cilobamine is an antidepressant and norepinephrine-dopamine reuptake inhibitor and has stimulant and antidepressant effects.

Chemical Structure

Cilobamine mesylate
Cilobamine mesylate
CAS#69429-85-2 (mesylate)

Theoretical Analysis

MedKoo Cat#: 412893

Name: Cilobamine mesylate

CAS#: 69429-85-2 (mesylate)

Chemical Formula: C18H27Cl2NO4S

Exact Mass: 0.0000

Molecular Weight: 424.38

Elemental Analysis: C, 50.94; H, 6.41; Cl, 16.71; N, 3.30; O, 15.08; S, 7.55

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Synonym
Cilobamine mesylate; Clobamine; RMI 81182EF; RMI-81182EF; RMI81182EF
IUPAC/Chemical Name
Bicyclo(2.2.2)octan-2-ol, 2-(3,4-dichlorophenyl)-3-((1-methylethyl)amino)-, cis-, methanesulfonate (salt)
InChi Key
VALAKNBZUXDQCX-YTOIOIGGSA-N
InChi Code
InChI=1S/C17H23Cl2NO.CH4O3S/c1-10(2)20-16-11-3-5-12(6-4-11)17(16,21)13-7-8-14(18)15(19)9-13;1-5(2,3)4/h7-12,16,20-21H,3-6H2,1-2H3;1H3,(H,2,3,4)/t11?,12?,16-,17-;/m1./s1
SMILES Code
O[C@@]1(C2=CC=C(Cl)C(Cl)=C2)C(CC3)CCC3[C@H]1NC(C)C.CS(=O)(O)=O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 424.38 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Leeson GA, Shaath ZA, Biedenbach SA, Yarrington JT, Okerholm RA. Dose related induction of the drug metabolizing enzymes of rat liver by cilobamine. Fundam Appl Toxicol. 1984 Apr;4(2 Pt 1):261-9. doi: 10.1016/0272-0590(84)90127-1. PMID: 6724198.