MedKoo Cat#: 412875 | Name: Ciclazindol hydrochloride

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Ciclazindol hydrochloride is the salt from of Ciclazindol (free base), a noradrenaline uptake inhibitor.

Chemical Structure

Ciclazindol hydrochloride
Ciclazindol hydrochloride
CAS#37647-67-9 (HCl)

Theoretical Analysis

MedKoo Cat#: 412875

Name: Ciclazindol hydrochloride

CAS#: 37647-67-9 (HCl)

Chemical Formula: C17H16Cl2N2O

Exact Mass:

Molecular Weight: 335.23

Elemental Analysis: C, 60.91; H, 4.81; Cl, 21.15; N, 8.36; O, 4.77

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Synonym
Ciclazindol hydrochloride; UNII-792OU8W6Z9
IUPAC/Chemical Name
Pyrimido(1,2-a)indol-10-ol, 10-(2-chlorophenyl)-2,3,4,10-tetrahydro-, hydrochloride (1:1)
InChi Key
VHYRNAQFPLEVJC-UHFFFAOYSA-N
InChi Code
InChI=1S/C17H15ClN2O.ClH/c18-14-8-3-1-6-12(14)17(21)13-7-2-4-9-15(13)20-11-5-10-19-16(17)20;/h1-4,6-9,21H,5,10-11H2;1H
SMILES Code
OC1(C2=CC=CC=C2Cl)C3=NCCCN3C4=C1C=CC=C4.[H]Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 335.23 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Kerr FA, Szabadi E. Comparison of the effects of chronic administration of ciclazindol and desipramine on pupillary responses to tyramine, methoxamine and pilocarpine in healthy volunteers. Br J Clin Pharmacol. 1985 May;19(5):639-47. doi: 10.1111/j.1365-2125.1985.tb02691.x. PMID: 4005103; PMCID: PMC1463841. 2: Ehsanullah RS, Kirby MJ, Leighton M, Oh VM. Some clinical pharmacological studies with ciclazindol hydrochloride [proceedings]. Br J Clin Pharmacol. 1977 Jun;4(3):400P. PMID: 901726. 3: Lean ME, Borthwick LJ. Ciclazindol: an oral agent with weight reducing properties and hypoglycaemic activity. Eur J Clin Pharmacol. 1983;25(1):41-5. doi: 10.1007/BF00544012. PMID: 6352281.