S1R-IN-10 is a novel selective sigma 1 receptor (S1R) antagonist, exhibiting potent binding affinity for S1R, high selectivity over S2R and 87 other human targets, acceptable in vitro metabolic stability, slowing clearance in liver microsomes, and excellent blood-brain barrier permeability in rats.
MedKoo Cat#: 463724
Name: S1R-IN-10
CAS#: unknown
Chemical Formula: C18H26N4
Exact Mass: 298.2157
Molecular Weight: 298.43
Elemental Analysis: C, 72.44; H, 8.78; N, 18.77
The following data is based on the product molecular weight 298.43 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
