Synonym
Carpronium (free base); UNII-X6UK728GLZ
IUPAC/Chemical Name
Ammonium, (3-carboxypropyl)trimethyl-, methyl ester
InChi Key
XQSLKIBWQSTAGK-UHFFFAOYSA-N
InChi Code
InChI=1S/C8H18NO2/c1-9(2,3)7-5-6-8(10)11-4/h5-7H2,1-4H3/q+1
SMILES Code
C[N+](C)(CCCC(OC)=O)C
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
Preparing Stock Solutions
The following data is based on the
product
molecular weight
160.24
Batch specific molecular weights may vary
from batch to batch
due to the degree of hydration, which will
affect the solvent
volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass |
1 mg |
5 mg |
10 mg |
| 1 mM |
1.15 mL |
5.76 mL |
11.51 mL |
| 5 mM |
0.23 mL |
1.15 mL |
2.3 mL |
| 10 mM |
0.12 mL |
0.58 mL |
1.15 mL |
| 50 mM |
0.02 mL |
0.12 mL |
0.23 mL |
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6: Ishida H, Mitsui K, Nukaya H, Matsumoto K, Tsuji K. Study of active substances involved in skin dysfunction induced by crowding stress. I. Effect of crowding and isolation on some physiological variables, skin function and skin blood perfusion in hairless mice. Biol Pharm Bull. 2003 Feb;26(2):170-81. doi: 10.1248/bpb.26.170. PMID: 12576676.
7: Shiraishi T. Effects of the non-amphetaminergic anorexiant, mazindol, on neuronal activity and hypothalamic control of gastric acid secretion in rats. Int J Obes. 1985;9(4):285-97. PMID: 3905642.
8: Morita K, Nakamura M, Nagamachi M, Kishi T, Miyachi Y. Seventeen cases of alopecia areata: combination of SADBE topical immunotherapy with other therapies. J Dermatol. 2002 Oct;29(10):661-4. doi: 10.1111/j.1346-8138.2002.tb00199.x. PMID: 12433000.
9: Shiraishi T. [Mazindol effects on the salivary and gastric acid secretory mechanisms]. Nihon Yakurigaku Zasshi. 1984 Feb;83(2):159-72. Japanese. PMID: 6745806.
10: Uchida T, Yamashita S. Purification and properties of choline kinase from rat brain. Biochim Biophys Acta. 1990 Apr 17;1043(3):281-8. doi: 10.1016/0005-2760(90)90028-v. PMID: 2157491.
