Methopholine is an opioid analgesic drug and isoquinoline derivative. Although it is not structurally related to most other opioids, Methopholine has around the analgesic activity as codeine and was evaluated for the treatment of postoperative pain. Metofoline tablets were marketed in the United States under the brand name of Versidyne, but the drug was withdrawn from the market in 1965 due to the occurrence of ophthalmic side-effects alongside the discovery that the drug could produce cataracts in dogs. NOT FOR INDIVIDUAL OR HUMAN USE.
MedKoo Cat#: 574985
Name: Methopholine
CAS#: 2154-02-1
Chemical Formula: C20H24ClNO2
Exact Mass: 345.1496
Molecular Weight: 345.87
Elemental Analysis: C, 69.45; H, 6.99; Cl, 10.25; N, 4.05; O, 9.25
The following data is based on the product molecular weight 345.87 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |