Cyclomethycaine | CAS # 139-62-8 | local anesthetic

MedKoo Cat#: 412224 | Name: Cyclomethycaine

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Cyclomethycaine is a local anesthetic

Chemical Structure

Cyclomethycaine

CAS#139-62-8

Theoretical Analysis

MedKoo Cat#: 412224

Name: Cyclomethycaine

CAS#: 139-62-8

Chemical Formula: C22H32NO3

Exact Mass: 358.2388

Molecular Weight: 358.50

Elemental Analysis: C, 73.71; H, 9.00; N, 3.91; O, 13.39

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

Cyclomethycaine; BRN-0293510; BRN0293510; BRN 0293510

IUPAC/Chemical Name

3-(2-Methylpiperidino)propyl-p-cyclohexyloxybenzoate

InChi Key

UCJGSYLTWJXITP-UHFFFAOYSA-M

InChi Code

InChI=1S/C22H33NO3/c1-17-8-5-6-14-23(17)15-7-9-18-16-19(22(24)25)12-13-21(18)26-20-10-3-2-4-11-20/h12-13,16-17,20H,2-11,14-15H2,1H3,(H,24,25)/p-1

SMILES Code

O=C([O-])C1=CC=C(OC2CCCCC2)C(CCCN3C(C)CCCC3)=C1

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 358.50 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Dorris RL. A comparison in rat and mouse heart of the ability of several local anesthetics to inhibit monoamine oxidase. Comp Biochem Physiol C Comp Pharmacol Toxicol. 1983;75(2):327-8. doi: 10.1016/0742-8413(83)90200-1. PMID: 6138200. 2: Fisher AA. Allergic reactions to topical (surface) anesthetics with reference to the safety of tronothane (pramoxine hydrochloride). Cutis. 1980 Jun;25(6):584, 586, 589-91 passim. PMID: 7379587. 3: Sciarra JJ, Patel SP. In vitro release of therapeutically active ingredients from polymer matrixes. J Pharm Sci. 1976 Oct;65(10):1519-22. doi: 10.1002/jps.2600651025. PMID: 978414. 4: Rabinovitch M, DeStefano M. Cell to substrate adhesion and spreading: inhibition by cationic anesthetics. J Cell Physiol. 1975 Apr;85(2 Pt 1):189-93. doi: 10.1002/jcp.1040850205. PMID: 235555. 5: CYCLOMETHYCAINE sulfate. J Am Med Assoc. 1957 May 18;164(3):280. PMID: 13415978. 6: MARSHALL BM. Surfacaine as a urological anesthetic. Urol Cutaneous Rev. 1949 Feb;53(2):86. PMID: 18108816.