MedKoo Cat#: 462813 | Name: U-32,802A

Description:

WARNING: This product is for research use only, not for human or veterinary use.

U-32,802A is a butyrophenone derivative that was found to block the uptake of and to cause a release of 3H-norepinephrine from the mouse heart.

Chemical Structure

U-32,802A
U-32,802A
CAS#36735-48-5

Theoretical Analysis

MedKoo Cat#: 462813

Name: U-32,802A

CAS#: 36735-48-5

Chemical Formula: C22H24ClF2NO

Exact Mass: 391.1514

Molecular Weight: 391.89

Elemental Analysis: C, 67.43; H, 6.17; Cl, 9.05; F, 9.70; N, 3.57; O, 4.08

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
No Data
Synonym
U 32802A; U32802A; U-32802A;
IUPAC/Chemical Name
4-((4'-fluoro-2,3,4,5-tetrahydro-[1,1'-biphenyl]-4-yl)amino)-1-(4-fluorophenyl)butan-1-one hydrochloride
InChi Key
HWSBEFRRYZIENO-UHFFFAOYSA-N
InChi Code
InChI=1S/C22H23F2NO.ClH/c23-19-9-3-16(4-10-19)17-7-13-21(14-8-17)25-15-1-2-22(26)18-5-11-20(24)12-6-18;/h3-7,9-12,21,25H,1-2,8,13-15H2;1H
SMILES Code
Fc1ccc(C(CCCNC2CCC(c3ccc(F)cc3)=CC2)=O)cc1.Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 391.89 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Lahti RA, Lednicer D. Effect of a butyrophenone derivative, U-32,802A, on brain biogenic amines. Biochem Pharmacol. 1974 Jun 15;23(12):1701-5. doi: 10.1016/0006-2952(74)90397-9. PMID: 4842658. 2: Fuenmayor LD, Vogt M. The influence of cerebral 5-hydroxytryptamine on catalepsy induced by brain-amine depleting neuroleptics or by cholinomimetics. Br J Pharmacol. 1979 Oct;67(2):309-18. doi: 10.1111/j.1476-5381.1979.tb08681.x. PMID: 40649; PMCID: PMC2043889. 3: Fuenmayor LD, Vogt M. Production of catalepsy and depletion of brain monoamines by a butyrophenone derivative. Br J Pharmacol. 1979 Sep;67(1):115-22. PMID: 574039; PMCID: PMC2043615.