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MedKoo Cat#: 573862 | Name: Amixetrine free base

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Amixetrine, also known as CERM 898; is said to be an anti-inflammatory, antidepressant, antispasmodic, anticholinergic, antihistamine, and antiserotonergic, but its definitive indications and pharmacology are unclear.

Chemical Structure

Amixetrine free base
Amixetrine free base
CAS#24622-72-8 (free base)

Theoretical Analysis

MedKoo Cat#: 573862

Name: Amixetrine free base

CAS#: 24622-72-8 (free base)

Chemical Formula: C17H27NO

Exact Mass: 261.2093

Molecular Weight: 261.41

Elemental Analysis: C, 78.11; H, 10.41; N, 5.36; O, 6.12

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
24622-52-4 (HCl) 24622-72-8 (free base)
Synonym
Amixetrine, CERM 898; CERM-898; CERM898;
IUPAC/Chemical Name
1-(beta-(Isopentyloxy)phenethyl)pyrrolidine
InChi Key
ISRODTBNJUAWEJ-UHFFFAOYSA-N
InChi Code
1S/C17H27NO/c1-15(2)10-13-19-17(14-18-11-6-7-12-18)16-8-4-3-5-9-16/h3-5,8-9,15,17H,6-7,10-14H2,1-2H3
SMILES Code
CC(C)CCOC(C1=CC=CC=C1)CN2CCCC2
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 261.41 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Constantin M, Pognat JF. Pharmacokinetics of amixetrine in the dog. Relation of dose-to-plasma concentration. Arzneimittelforschung. 1978;28(4):646-51. PubMed PMID: 581941. 2: André C, Lambert R, Fargier MC. [A double-blind endoscopic, histologic and immunohistochemical study of the effect of amixetrine in the treatment of antritis (author's transl)]. Biol Gastroenterol (Paris). 1976 Oct-Nov;9(4):283-8. French. PubMed PMID: 798603. 3: Constatin M, Pognat JF, Streichenberger G. Urinary metabolites of amixetrine in man and in the dog. Arzneimittelforschung. 1976;26(1):80-7. PubMed PMID: 947187.