MedKoo Cat#: 565481 | Name: ElteN378
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

ElteN378 is a novel potent fkbp12 ligand

Chemical Structure

ElteN378
ElteN378
CAS#1421366-99-5

Theoretical Analysis

MedKoo Cat#: 565481

Name: ElteN378

CAS#: 1421366-99-5

Chemical Formula: C23H26N2O3

Exact Mass: 378.1943

Molecular Weight: 378.47

Elemental Analysis: C, 72.99; H, 6.92; N, 7.40; O, 12.68

Price and Availability

Size Price Availability Quantity
25mg USD 950.00 2 Weeks
50mg USD 1,650.00 2 Weeks
100mg USD 2,450.00 2 Weeks
1g USD 5,450.00 2 Weeks
2g USD 8,650.00 2 Weeks
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Related CAS #
No Data
Synonym
ElteN378; Elte N378; Elte-N378
IUPAC/Chemical Name
(S)-1-(2-Oxo-2-phenylacetyl)-N-(3-phenylpropyl)piperidine-2-carboxamide
InChi Key
QXYDCLICGYMGIX-FQEVSTJZSA-N
InChi Code
InChI=1S/C23H26N2O3/c26-21(19-13-5-2-6-14-19)23(28)25-17-8-7-15-20(25)22(27)24-16-9-12-18-10-3-1-4-11-18/h1-6,10-11,13-14,20H,7-9,12,15-17H2,(H,24,27)/t20-/m0/s1
SMILES Code
O=C([C@H]1N(C(C(C2=CC=CC=C2)=O)=O)CCCC1)NCCCC3=CC=CC=C3
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 378.47 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Martina MR, Tenori E, Bizzarri M, Menichetti S, Caminati G, Procacci P. The precise chemical-physical nature of the pharmacore in FK506 binding protein inhibition: ElteX, a New class of nanomolar FKBP12 ligands. J Med Chem. 2013 Feb 14;56(3):1041-51. doi: 10.1021/jm3015052. Epub 2013 Jan 24. PubMed PMID: 23301792.