GSK2643943A is a potent USP20 inhibitor with IC50 = 160 nM.
MedKoo Cat#: 555407
Name: GSK2643943A
CAS#: 2449301-27-1 (free base)
Chemical Formula: C17H12FN3
Exact Mass: 277.1015
Molecular Weight: 277.30
Elemental Analysis: C, 73.63; H, 4.36; F, 6.85; N, 15.15
| Solvent | mg/mL | mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 90.0 | 324.56 | |
| Ethanol | 8.0 | 28.85 |
The following data is based on the product molecular weight 277.30 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
