Propyromazine bromide | CAS#145-54-0 | Anticholinergic

MedKoo Cat#: 598510 | Name: Propyromazine bromide

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Propyromazine bromide is a quatemary ammonium with muscarinic cholinoceptor antagonistic activity. This antimuscarinic agent with peripheral effects similar to those of atropine is given in the symptomatic treatment of visceral spasm.

Chemical Structure

Propyromazine bromide

CAS#145-54-0

Theoretical Analysis

MedKoo Cat#: 598510

Name: Propyromazine bromide

CAS#: 145-54-0

Chemical Formula: C20H23BrN2OS

Exact Mass: 0.0000

Molecular Weight: 419.38

Elemental Analysis: C, 57.28; H, 5.53; Br, 19.05; N, 6.68; O, 3.81; S, 7.64

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

Propyromazine bromide; Diospasmyl; LD 335; LD-335; LD335; NSC 169416; NSC-169416; NSC169416;

IUPAC/Chemical Name

1-methyl-1-(1-oxo-1-(10H-phenothiazin-10-yl)propan-2-yl)pyrrolidin-1-ium bromide

InChi Key

OANVFVBYPNXRLD-UHFFFAOYSA-M

InChi Code

InChI=1S/C20H23N2OS.BrH/c1-15(22(2)13-7-8-14-22)20(23)21-16-9-3-5-11-18(16)24-19-12-6-4-10-17(19)21;/h3-6,9-12,15H,7-8,13-14H2,1-2H3;1H/q+1;/p-1

SMILES Code

CC([N+]1(C)CCCC1)C(N2C3=C(C=CC=C3)SC4=CC=CC=C24)=O.[Br-]

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.03.00

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 419.38 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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