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MedKoo Cat#: 597468 | Name: Diallyl G

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Diallyl G is a delta-opioid receptor antagonist.

Chemical Structure

Diallyl G
CAS#127808-81-5

Theoretical Analysis

MedKoo Cat#: 597468

Name: Diallyl G

CAS#: 127808-81-5

Chemical Formula: C38H53N5O8

Exact Mass: 707.3894

Molecular Weight: 707.86

Elemental Analysis: C, 64.48; H, 7.55; N, 9.89; O, 18.08

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Diallyl G; Diallyl-G; DiallylG; N,N-Diallyl-tyr-D-leu-gly-tyr-leu-OH; N,N-Diallyl-tyrosyl-leucyl-glycyl-tyrosyl-leucine;
IUPAC/Chemical Name
diallyl-L-tyrosyl-D-leucylglycyl-L-tyrosyl-L-leucine
InChi Key
WPYLFYWRECLMCS-GJBCSVNNSA-N
InChi Code
InChI=1S/C38H53N5O8/c1-7-17-43(18-8-2)33(22-27-11-15-29(45)16-12-27)37(49)41-30(19-24(3)4)35(47)39-23-34(46)40-31(21-26-9-13-28(44)14-10-26)36(48)42-32(38(50)51)20-25(5)6/h7-16,24-25,30-33,44-45H,1-2,17-23H2,3-6H3,(H,39,47)(H,40,46)(H,41,49)(H,42,48)(H,50,51)/t30-,31+,32+,33+/m1/s1
SMILES Code
CC(C)C[C@@H](C(O)=O)NC([C@H](CC1=CC=C(O)C=C1)NC(CNC([C@@H](CC(C)C)NC([C@H](CC2=CC=C(O)C=C2)N(CC=C)CC=C)=O)=O)=O)=O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 707.86 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Georgoussi Z, Zioudrou C. Effect of delta-opioid antagonists on the functional coupling between opioid receptors and G-proteins in rat brain membranes. Biochem Pharmacol. 1993 Jun 22;45(12):2405-10. PubMed PMID: 8392341. 2: Dragatsis I, Zioudrou C, Gerozissis K. Specific delta-opioid antagonists exert an agonist-independent inhibitory effect, similar to the agonist, on the release of GnRH in vitro. Cell Mol Neurobiol. 1995 Aug;15(4):389-400. PubMed PMID: 8565043. 3: Gerozissis K, Dragatsis I, Zioudrou C. The delta-opioid signal transduction on the gonadotropin-releasing hormone release is eicosanoid dependent. Brain Res. 1993 Oct 29;626(1-2):219-24. PubMed PMID: 8281433. 4: Loukas S, Mercouris M, Panetsos F, Zioudrou C. Purification to homogeneity of an active opioid receptor from rat brain by affinity chromatography. Proc Natl Acad Sci U S A. 1994 May 10;91(10):4574-8. PubMed PMID: 8183950; PubMed Central PMCID: PMC43828. 5: Dragatsis I, Papazafiri P, Zioudrou C, Gerozissis K. Opioids modify the release of LH at the pituitary level: in vitro studies with entire rat pituitaries. J Endocrinol. 1995 May;145(2):263-70. PubMed PMID: 7616159.