Doxapram HCl hydrate | CAS# 7081-53-0 | Potassium Channel Inhibitor

MedKoo Cat#: 591486 | Name: Doxapram hydrochloride hydrate

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Description:

WARNING: This product is for research use only, not for human or veterinary use.

Doxapram hydrochloride (marketed as Dopram, Stimulex or Respiram) is a respiratory stimulant. Administered intravenously, doxapram stimulates an increase in tidal volume, and respiratory rate.

Chemical Structure

Doxapram hydrochloride hydrate

CAS#7081-53-0 (HCl hydrate)

Theoretical Analysis

MedKoo Cat#: 591486

Name: Doxapram hydrochloride hydrate

CAS#: 7081-53-0 (HCl hydrate)

Chemical Formula: C24H33ClN2O3

Exact Mass: 0.0000

Molecular Weight: 432.99

Elemental Analysis: C, 66.58; H, 7.68; Cl, 8.19; N, 6.47; O, 11.09

Price and Availability

Size	Price	Availability
25mg	USD 250.00	2 Weeks
50mg	USD 450.00	2 Weeks
100mg	USD 750.00	2 Weeks

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Related CAS #

309-29-5 (free base) 7081-53-0 (HCl hydrate)

Synonym

Doxapram hydrochloride monohydrate; Doxapram HCl hydrate; Dopram; AHR 619; AHR-619; AHR619

IUPAC/Chemical Name

2-Pyrrolidinone, 1-ethyl-4-(2-(4-morpholinyl)ethyl)-3,3-diphenyl-, monohydrochloride, monohydrate

InChi Key

ZOMBFZRWMLIDPX-UHFFFAOYSA-N

InChi Code

InChI=1S/C24H30N2O2.ClH.H2O/c1-2-26-19-22(13-14-25-15-17-28-18-16-25)24(23(26)27,20-9-5-3-6-10-20)21-11-7-4-8-12-21;;/h3-12,22H,2,13-19H2,1H3;1H;1H2

SMILES Code

O=C1N(CC)CC(CCN2CCOCC2)C1(C3=CC=CC=C3)C4=CC=CC=C4.[H]Cl.[H]O[H]

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Product Data

Product Data

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 432.99 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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