L-796568 free base is a β3 adrenergic receptor agonist potentially for the treatment of obesity. L-796568 is a potent full beta(3) agonist (EC(50) = 3.6 nM, 94% activation) with >600-fold selectivity over the human beta(1) and beta(2) receptors, which also displays good oral bioavailability in several mammalian species, as well as an extended duration of action.
MedKoo Cat#: 596705
Name: L-796568 free base
CAS#: 211031-01-5
Chemical Formula: C31H27F3N4O3S2
Exact Mass: 624.1477
Molecular Weight: 624.69
Elemental Analysis: C, 59.60; H, 4.36; F, 9.12; N, 8.97; O, 7.68; S, 10.26
The following data is based on the product molecular weight 624.69 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |