MedKoo Cat#: 341534 | Name: Cyprazepam

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Cyprazepam is a biochemical. This drug is unscheduled in the USA.

Chemical Structure

Cyprazepam
Cyprazepam
CAS#15687-07-7

Theoretical Analysis

MedKoo Cat#: 341534

Name: Cyprazepam

CAS#: 15687-07-7

Chemical Formula: C19H18ClN3O

Exact Mass:

Molecular Weight: 339.82

Elemental Analysis: C, 67.16; H, 5.34; Cl, 10.43; N, 12.37; O, 4.71

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
No Data
Synonym
Cyprazepam; W 3623; W-3623; W3623
IUPAC/Chemical Name
3H-1,4-Benzodiazepin-2-amine, 7-chloro-N-(cyclopropylmethyl)-5-phenyl-, 4-oxide
InChi Key
UKFDTMNJMKWWNK-UHFFFAOYSA-N
InChi Code
InChI=1S/C19H18ClN3O/c20-15-8-9-17-16(10-15)19(14-4-2-1-3-5-14)23(24)12-18(22-17)21-11-13-6-7-13/h1-5,8-10,13H,6-7,11-12H2,(H,21,22)
SMILES Code
ClC1=CC=C(N=C(NCC2CC2)C[N+]([O-])=C3C4=CC=CC=C4)C3=C1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 339.82 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Moretti M, Andrello L, Visonà S, Vignali C, Groppi A, Freni F, Osculati A, Tajana L, Morini L. Evaluation of benzodiazepines and zolpidem in nails and their stability after prolonged exposure to chlorinated water. J Pharm Biomed Anal. 2018 Apr 15;152:137-142. doi: 10.1016/j.jpba.2018.01.051. Epub 2018 Jan 31. PubMed PMID: 29414005. 2: Dinis-Oliveira RJ. Metabolic profile of oxazepam and related benzodiazepines: clinical and forensic aspects. Drug Metab Rev. 2017 Nov;49(4):451-463. doi: 10.1080/03602532.2017.1377223. Epub 2017 Sep 14. Review. PubMed PMID: 28903606. 3: Aknouche F, Guibert E, Tessier A, Eibel A, Kintz P. Suicide by ingestion of caffeine. Egypt J Forensic Sci. 2017;7(1):6. doi: 10.1186/s41935-017-0001-2. Epub 2017 Jul 19. PubMed PMID: 28781898; PubMed Central PMCID: PMC5514181. 4: De Boeck M, Missotten S, Dehaen W, Tytgat J, Cuypers E. Development and validation of a fast ionic liquid-based dispersive liquid-liquid microextraction procedure combined with LC-MS/MS analysis for the quantification of benzodiazepines and benzodiazepine-like hypnotics in whole blood. Forensic Sci Int. 2017 May;274:44-54. doi: 10.1016/j.forsciint.2016.12.026. Epub 2016 Dec 26. PubMed PMID: 28094153. 5: Bénard-Laribière A, Noize P, Pambrun E, Bazin F, Verdoux H, Tournier M, Bégaud B, Pariente A. Trends in incident use of benzodiazepines and Z-drugs in France from 2006 to 2012: a population-based study. Pharmacoepidemiol Drug Saf. 2017 Feb;26(2):162-169. doi: 10.1002/pds.4123. Epub 2016 Nov 3. PubMed PMID: 27807907. 6: Potocka-Banaś B, Dembińska T, Borowiak K. [Benzodiazepines’ reactivity in immunoassay techniques – problems with interpretation]. Pomeranian J Life Sci. 2016;62(3):21-6. Polish. PubMed PMID: 29537762. 7: Cloos JM, Bocquet V, Rolland-Portal I, Koch P, Chouinard G. Hypnotics and Triazolobenzodiazepines--Best Predictors of High-Dose Benzodiazepine Use: Results from the Luxembourg National Health Insurance Registry. Psychother Psychosom. 2015;84(5):273-83. doi: 10.1159/000434755. Epub 2015 Aug 6. PubMed PMID: 26278327. 8: Hahirwa I, Charlier C, Karangwa C, Denooz R. Determination of blood concentration levels of psychotropic medications in Rwandan patients. Acta Clin Belg. 2015 Dec;70(6):425-31. doi: 10.1179/2295333715Y.0000000055. Epub 2015 Jul 28. PubMed PMID: 26220264. 9: de Beaurepaire R, Trinh I, Guirao S, Taieb M. Colitis possibly induced by quetiapine. BMJ Case Rep. 2015 Feb 26;2015. pii: bcr2014207912. doi: 10.1136/bcr-2014-207912. PubMed PMID: 25721830; PubMed Central PMCID: PMC4342667. 10: Sabia R, Ciogli A, Pierini M, Gasparrini F, Villani C. Dynamic high performance liquid chromatography on chiral stationary phases. Low temperature separation of the interconverting enantiomers of diazepam, flunitrazepam, prazepam and tetrazepam. J Chromatogr A. 2014 Oct 10;1363:144-9. doi: 10.1016/j.chroma.2014.07.097. Epub 2014 Aug 12. PubMed PMID: 25138707. 11: Toubou H, Namera A, Arima Y, Uchida Y, Torikoshi A, Moriya F, Nagao M. Detection of abused drugs in human blood by using the on-site drug-screening device Oratect® III. Leg Med (Tokyo). 2014 Sep;16(5):308-13. doi: 10.1016/j.legalmed.2014.04.004. Epub 2014 May 9. PubMed PMID: 24877596. 12: Guarneri F, Guarneri C, Marini H. Oral lichen planus and neurogenic inflammation: new observations and therapeutic implications from four clinical cases. Dermatol Ther. 2014 Jul-Aug;27(4):206-10. doi: 10.1111/dth.12118. Epub 2014 Feb 18. PubMed PMID: 24548522. 13: Kumari S, Mohana Priya A, Lulu S, Tauqueer M. Molecular modeling, simulation and virtual screening of ribosomal phosphoprotein P1 from Plasmodium falciparum. J Theor Biol. 2014 Feb 21;343:113-9. doi: 10.1016/j.jtbi.2013.10.014. Epub 2013 Nov 7. Erratum in: J Theor Biol. 2014 Aug 7;354:146. PubMed PMID: 24211527. 14: Altamura AC, Moliterno D, Paletta S, Maffini M, Mauri MC, Bareggi S. Understanding the pharmacokinetics of anxiolytic drugs. Expert Opin Drug Metab Toxicol. 2013 Apr;9(4):423-40. doi: 10.1517/17425255.2013.759209. Epub 2013 Jan 21. Review. PubMed PMID: 23330992. 15: Verplaetse R, Cuypers E, Tytgat J. The evaluation of the applicability of a high pH mobile phase in ultrahigh performance liquid chromatography tandem mass spectrometry analysis of benzodiazepines and benzodiazepine-like hypnotics in urine and blood. J Chromatogr A. 2012 Aug 3;1249:147-54. doi: 10.1016/j.chroma.2012.06.023. Epub 2012 Jun 15. PubMed PMID: 22749457. 16: Richards BL, Whittle SL, Buchbinder R. Muscle relaxants for pain management in rheumatoid arthritis. Cochrane Database Syst Rev. 2012 Jan 18;1:CD008922. doi: 10.1002/14651858.CD008922.pub2. Review. PubMed PMID: 22258993. 17: Rust KY, Baumgartner MR, Meggiolaro N, Kraemer T. Detection and validated quantification of 21 benzodiazepines and 3 "z-drugs" in human hair by LC-MS/MS. Forensic Sci Int. 2012 Feb 10;215(1-3):64-72. doi: 10.1016/j.forsciint.2011.07.052. Epub 2011 Aug 27. PubMed PMID: 21873006. 18: Chavant F, Favrelière S, Lafay-Chebassier C, Plazanet C, Pérault-Pochat MC. Memory disorders associated with consumption of drugs: updating through a case/noncase study in the French PharmacoVigilance Database. Br J Clin Pharmacol. 2011 Dec;72(6):898-904. doi: 10.1111/j.1365-2125.2011.04009.x. PubMed PMID: 21557759; PubMed Central PMCID: PMC3244635. 19: Rossat A, Fantino B, Bongue B, Colvez A, Nitenberg C, Annweiler C, Beauchet O. Association between benzodiazepines and recurrent falls: a cross-sectional elderly population-based study. J Nutr Health Aging. 2011 Jan;15(1):72-7. PubMed PMID: 21267523. 20: Hayase N, Iwayama K, Ohtaki K, Yamashita Y, Awaya T, Matsubara K. [Dissolution behaviors of tablet and capsule covered with oblate or agar jelly for taking medicine easily]. Yakugaku Zasshi. 2011 Jan;131(1):161-8. Japanese. PubMed PMID: 21212625.