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MedKoo Cat#: 581173 | Name: Dacemazine

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Dacemazine is used in treatment of Depression.

Chemical Structure

Dacemazine
Dacemazine
CAS#518-61-6

Theoretical Analysis

MedKoo Cat#: 581173

Name: Dacemazine

CAS#: 518-61-6

Chemical Formula: C16H16N2OS

Exact Mass: 284.0983

Molecular Weight: 284.38

Elemental Analysis: C, 67.58; H, 5.67; N, 9.85; O, 5.63; S, 11.27

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
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Synonym
Dacemazine; Ahistan; BRN 0027765; Dacemazinum; Dimethylglycylphenothiazine; Histantin richter;
IUPAC/Chemical Name
10-((Dimethylamino)acetyl)-10H-phenothiazine
InChi Key
HKUCYAHWPVLPFN-UHFFFAOYSA-N
InChi Code
InChI=1S/C16H16N2OS/c1-17(2)11-16(19)18-12-7-3-5-9-14(12)20-15-10-6-4-8-13(15)18/h3-10H,11H2,1-2H3
SMILES Code
O=C(N1C2=C(C=CC=C2)SC3=CC=CC=C13)CN(C)C
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 284.38 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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Nutr Cancer. 2016 Jul;68(5):811-7. doi: 10.1080/01635581.2016.1170167. Epub 2016 May 13. PubMed PMID: 27176572. 10: Kansal S, Negi AK, Bhatnagar A, Agnihotri N. Ras signaling pathway in the chemopreventive action of different ratios of fish oil and corn oil in experimentally induced colon carcinogenesis. Nutr Cancer. 2012;64(4):559-68. doi: 10.1080/01635581.2012.675619. Epub 2012 Apr 20. PubMed PMID: 22519408. 11: Poulsen M, Mortensen A, Binderup ML, Langkilde S, Markowski J, Dragsted LO. The effect of apple feeding on markers of colon carcinogenesis. Nutr Cancer. 2011;63(3):402-9. doi: 10.1080/01635581.2011.535961. PubMed PMID: 21432724. 12: 1,1-Dimethylhydrazine. IARC Monogr Eval Carcinog Risks Hum. 1999;71 Pt 3:1425-36. Review. PubMed PMID: 10476423. 13: Lovinskaya AV, Kolumbayeva SZh, Abilev SK, Kolomiets OL. [IMMUNOCYTOCHEMICAL ANALYSIS OF THE DISTURBANCES IN THE STRUCTURE OF SYNAPTONEMAL COMPLEXES IN SPERMATOCYTE NUCLEI IN MICE UNDER EXPOSURE TO ROCKET FUEL COMPONENT]. 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