DCG066 is a G9a inhibitor. DCG066 can bind directly to G9a and inhibit methyltransferase activity in vitro. It displays low cytotoxicity in leukemia cell lines with high levels of G9a expression, including K562.
MedKoo Cat#: 561309
Name: DCG066
CAS#: 494786-13-9
Chemical Formula: C30H31F6N3O2
Exact Mass: 579.2320
Molecular Weight: 579.59
Elemental Analysis: C, 62.17; H, 5.39; F, 19.67; N, 7.25; O, 5.52
The following data is based on the product molecular weight 579.59 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
