LDN-0212320 Maleate | EAAT2 translation | CAS#894002-50-7

MedKoo Cat#: 525692 | Name: LDN-0212320 Maleate

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Description:

WARNING: This product is for research use only, not for human or veterinary use.

LDN-0212320 Maleate is a novel activator of glutamate transporter EAAT2 translation.

Chemical Structure

LDN-0212320 Maleate

CAS#894002-50-7

Theoretical Analysis

MedKoo Cat#: 525692

Name: LDN-0212320 Maleate

CAS#: 894002-50-7

Chemical Formula: C21H19N3O4S

Exact Mass: 0.0000

Molecular Weight: 409.46

Elemental Analysis: C, 61.60; H, 4.68; N, 10.26; O, 15.63; S, 7.83

Price and Availability

Size	Price	Availability
10mg	USD 450.00	2 Weeks
25mg	USD 750.00	2 Weeks
50mg	USD 1,050.00	2 Weeks

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Related CAS #

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Synonym

LDN-0212320 Maleate; LDN0212320; LDN 0212320

IUPAC/Chemical Name

3-[[(2-Methylphenyl)methyl]thio]-6-(2-pyridinyl)-pyridazine maleate

InChi Key

QIGJQEQXFAVIPF-BTJKTKAUSA-N

InChi Code

InChI=1S/C17H15N3S.C4H4O4/c1-13-6-2-3-7-14(13)12-21-17-10-9-16(19-20-17)15-8-4-5-11-18-15;5-3(6)1-2-4(7)8/h2-11H,12H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-

SMILES Code

CC1=CC=CC=C1CSC2=NN=C(C3=NC=CC=C3)C=C2.O=C(O)/C=C\C(O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 409.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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