RS 39604 HCl is a potent and selective 5-HT4 antagonist, with a pKi of 9.1 at 5-HT4 receptors in guinea pig striatal membranes and greater than 1000-fold selectivity over 5-HT1A, 2C, 3 and D1, D2, M1, M2, AT1, B1 and α1C receptors.
MedKoo Cat#: 532589
Name: RS 39604 HCl
CAS#: 167710-87-4(RS 39604 HCl); 172679-58-2(RS 39604).
Chemical Formula: C16H24Cl2N2O3
Exact Mass:
Molecular Weight: 363.28
Elemental Analysis: C, 52.90; H, 6.66; Cl, 19.52; N, 7.71; O, 13.21
The following data is based on the product molecular weight 363.28 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
