PG 01037 dihydrochloride is a dopamine D3 receptor antagonist. PG 01037 dihydrochloride is 133-fold selective for D3 over D2 receptors in vitro (Ki values are 0.70, 93.3 and 375 nM for D3, D2 and D4 receptors respectively).
MedKoo Cat#: 532469
Name: PG 01037 dihydrochloride
CAS#: 675599-62-9 (HCl)
Chemical Formula: C26H28Cl4N4O
Exact Mass: 0.0000
Molecular Weight: 554.34
Elemental Analysis: C, 56.34; H, 5.09; Cl, 25.58; N, 10.11; O, 2.89
The following data is based on the product molecular weight 554.34 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
