MedKoo Cat#: 531748 | Name: CP 93129 Dihydrochloride
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

CP 93129 Dihydrochloride is a 5HT(1B) receptor agonist. In rodent globus pallidus (GP) CP 93129 dihydrochloride could reduce GABA release in vitro and reverse reserpine-induced akinesia in vivo.

Chemical Structure

CP 93129 Dihydrochloride
CP 93129 Dihydrochloride
CAS#879089-64-2 (2HCl)

Theoretical Analysis

MedKoo Cat#: 531748

Name: CP 93129 Dihydrochloride

CAS#: 879089-64-2 (2HCl)

Chemical Formula: C12H15Cl2N3O

Exact Mass: 0.0000

Molecular Weight: 288.17

Elemental Analysis: C, 50.02; H, 5.25; Cl, 24.60; N, 14.58; O, 5.55

Price and Availability

Size Price Availability Quantity
10mg USD 450.00 2 Weeks
25mg USD 850.00 2 Weeks
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Synonym
CP 93129 Dihydrochloride; CP 93129 2HCl; CP 93129; CP93129; CP-93129.
IUPAC/Chemical Name
1,4-Dihydro-3-(1,2,3,6-tetrahydro-4-pyridinyl)-5H-pyrrol[3,2-b]pyridin-5-one dihydrochloride
InChi Key
FLVJHUZZKVJQNH-UHFFFAOYSA-N
InChi Code
InChI=1S/C12H13N3O.2ClH/c16-11-2-1-10-12(15-11)9(7-14-10)8-3-5-13-6-4-8;;/h1-3,7,13-14H,4-6H2,(H,15,16);2*1H
SMILES Code
O=C1C=CC(NC=C2C3=CCNCC3)=C2N1.[H]Cl.[H]Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 288.17 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Chadha A, Sur C, Atack J, Duty S. The 5HT(1B) receptor agonist, CP-93129, inhibits [(3)H]-GABA release from rat globus pallidus slices and reverses akinesia following intrapallidal injection in the reserpine-treated rat. Br J Pharmacol. 2000 Aug;130(8):1927-32. PubMed PMID: 10952684; PubMed Central PMCID: PMC1572281.