Veledimex | CAS#1093130-72-3

MedKoo Cat#: 529812 | Name: Veledimex

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Veledimex, also known as AD-1001, INXN-1001 and RG-115932 is a drug potentially for the treatment of melanoma and breast cancer

Chemical Structure

Veledimex

CAS#1093130-72-3

Theoretical Analysis

MedKoo Cat#: 529812

Name: Veledimex

CAS#: 1093130-72-3

Chemical Formula: C27H38N2O3

Exact Mass: 438.2882

Molecular Weight: 438.61

Elemental Analysis: C, 73.94; H, 8.73; N, 6.39; O, 10.94

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

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Related CAS #

1093130-72-3

Synonym

AD-1001; AD1001; AD 1001; INXN-1001;INXN1001; INXN 1001; RG-115932; RG115932; RG 115932; Veledimex.

IUPAC/Chemical Name

(R)-N'-(3,5-dimethylbenzoyl)-N'-(2,2-dimethylhexan-3-yl)-2-ethyl-3-methoxybenzohydrazide

InChi Key

LZWZPGLVHLSWQX-XMMPIXPASA-N

InChi Code

InChI=1S/C27H38N2O3/c1-9-12-24(27(5,6)7)29(26(31)20-16-18(3)15-19(4)17-20)28-25(30)22-13-11-14-23(32-8)21(22)10-2/h11,13-17,24H,9-10,12H2,1-8H3,(H,28,30)/t24-/m1/s1

SMILES Code

O=C(NN(C(C1=CC(C)=CC(C)=C1)=O)[C@@H](C(C)(C)C)CCC)C2=CC=CC(OC)=C2CC

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 438.61 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Cai H, Sun L, Miao J, Krishman S, Lebel F, Barrett JA. Plasma Pharmacokinetics of Veledimex, a Small-Molecule Activator Ligand for a Proprietary Gene Therapy Promoter System, in Healthy Subjects. Clin Pharmacol Drug Dev. 2016 Jul 1. doi: 10.1002/cpdd.287. [Epub ahead of print] PubMed PMID: 27364771.