MedKoo Cat#: 524686 | Name: Cgp 29030A

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Cgp 29030A is a novel piperazine derivative that has marked inhibitory action on presumably nociceptive dorsal horn neurons that processed input from high-threshold mechanosensitive receptors in the skin and deep somatic tissues (muscle, tendon, joint). It may be of benefit in the treatment of painful disorders which are complicated by increased motor activity.

Chemical Structure

Cgp 29030A
Cgp 29030A
CAS#113240-27-0

Theoretical Analysis

MedKoo Cat#: 524686

Name: Cgp 29030A

CAS#: 113240-27-0

Chemical Formula: C21H26Cl2N2O3

Exact Mass:

Molecular Weight: 425.35

Elemental Analysis: C, 59.30; H, 6.16; Cl, 16.67; N, 6.59; O, 11.28

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Cgp 29030A; Cgp29030A; Cgp-29030A.
IUPAC/Chemical Name
Piperazine, 1-(2-(4-chlorophenyl)ethyl)-4-(3,5-dimethoxybenzoyl)-, monohydrochloride
InChi Key
OGLXGFIBROXFPU-UHFFFAOYSA-N
InChi Code
InChI=1S/C21H25ClN2O3.ClH/c1-26-19-13-17(14-20(15-19)27-2)21(25)24-11-9-23(10-12-24)8-7-16-3-5-18(22)6-4-16;/h3-6,13-15H,7-12H2,1-2H3;1H
SMILES Code
COc1cc(cc(c1)OC)C(=O)N2CCN(CC2)CCc3ccc(cc3)Cl.Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO, not in water
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 425.35 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Yu XM, Hoheisel U, Mense S. Effects of a novel piperazine derivative (CGP 29030A) on nociceptive dorsal horn neurons in the rat. Drugs Exp Clin Res. 1992;18(11-12):447-59. PubMed PMID: 1308469.