PD-224378 | CAS#466678-44-4 | biochemical

MedKoo Cat#: 145696 | Name: PD-224378

Description:

WARNING: This product is for research use only, not for human or veterinary use.

PD-224378 is a chemical compound that acts as a selective antagonist of the dopamine D4 receptor. It has been primarily studied in the context of neuroscience and pharmacology, as dopamine receptors play a key role in various brain functions, including mood, cognition, and movement.

Chemical Structure

PD-224378

CAS#466678-44-4

Theoretical Analysis

MedKoo Cat#: 145696

Name: PD-224378

CAS#: 466678-44-4

Chemical Formula: C20H35NO11

Exact Mass: 465.2200

Molecular Weight: 465.50

Elemental Analysis: C, 51.61; H, 7.58; N, 3.01; O, 37.81

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

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Related CAS #

No Data

Synonym

PD-224378;

IUPAC/Chemical Name

(S)-1-((2R,3R,4R,5S,6R)-3,4-dihydroxy-6-(hydroxymethyl)-5-(((2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)oxy)tetrahydro-2H-pyran-2-yl)-4-isobutylpyrrolidin-2-one

InChi Key

BSKMCHXCKWARJQ-PZXPMIFTSA-N

InChi Code

1S/C20H35NO11/c1-8(2)3-9-4-12(24)21(5-9)19-16(28)15(27)18(11(7-23)30-19)32-20-17(29)14(26)13(25)10(6-22)31-20/h8-11,13-20,22-23,25-29H,3-7H2,1-2H3/t9-,10+,11+,13-,14-,15+,16+,17+,18+,19+,20-/m0/s1

SMILES Code

[H][C@@]3(O[C@@H]1[C@@H](CO)O[C@H]([C@H](O)[C@H]1O)N2C[C@@H](CC(C)C)CC2=O)O[C@H](CO)[C@H](O)[C@H](O)[C@H]3O

Appearance

To be determined

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 465.50 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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