MedKoo Cat#: 128267 | Name: GLP-1R agonist DMB
Featured

Description:

WARNING: This product is for research use only, not for human or veterinary use.

GLP-1R agonist 2 (compound 2) is an effective GLP-1R agonist that exerts its activating effect by forming hydrogen bonds with the Tyr42, Cys71, and Ser84 residues of GLP-1R.

Chemical Structure

GLP-1R agonist DMB
GLP-1R agonist DMB
CAS#281209-71-0

Theoretical Analysis

MedKoo Cat#: 128267

Name: GLP-1R agonist DMB

CAS#: 281209-71-0

Chemical Formula: C13H15Cl2N3O2S

Exact Mass: 347.0262

Molecular Weight: 348.24

Elemental Analysis: C, 44.84; H, 4.34; Cl, 20.36; N, 12.07; O, 9.19; S, 9.21

Price and Availability

Size Price Availability Quantity
10mg USD 350.00 2 Weeks
25mg USD 650.00 2 Weeks
50mg USD 950.00 2 Weeks
Bulk Inquiry
Buy Now
Add to Cart
Related CAS #
No Data
Synonym
GLP-1R agonist DMB; GLP1R agonist DMB; GLP 1R agonist DMB
IUPAC/Chemical Name
N-(tert-butyl)-6,7-dichloro-3-(methylsulfonyl)quinoxalin-2-amine
InChi Key
GNZCSGYHILBXLL-UHFFFAOYSA-N
InChi Code
InChI=1S/C13H15Cl2N3O2S/c1-13(2,3)18-11-12(21(4,19)20)17-10-6-8(15)7(14)5-9(10)16-11/h5-6H,1-4H3,(H,16,18)
SMILES Code
O=S(C1=NC2=CC(Cl)=C(Cl)C=C2N=C1NC(C)(C)C)(C)=O
Appearance
To be determined
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 348.24 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Girdhar K, Dehury B, Kumar Singh M, Daniel VP, Choubey A, Dogra S, Kumar S, Mondal P. Novel insights into the dynamics behavior of glucagon-like peptide-1 receptor with its small molecule agonists. J Biomol Struct Dyn. 2019 Sep;37(15):3976-3986. doi: 10.1080/07391102.2018.1532818. Epub 2018 Nov 17. PMID: 30296922.