YZ-202 is a free-acid form of orbofiban. YZ202 is classified as a class II GPIIb/IIIa antagonist and demonstrates comparable antiaggregatory efficacy but lower potency in altering the strength of TF-mediated clot formation compared to class I antagonists, such as XV459 and DMP802, suggesting a differential effect on platelet-fibrin clot retraction despite similar antiaggregatory potency.
MedKoo Cat#: 145055
Name: YZ-202
CAS#: 199530-77-3
Chemical Formula: C15H19N5O4
Exact Mass: 333.1437
Molecular Weight: 333.35
Elemental Analysis: C, 54.05; H, 5.75; N, 21.01; O, 19.20
The following data is based on the product molecular weight 333.35 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
