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MedKoo Cat#: 125654 | Name: LUF5484

Description:

WARNING: This product is for research use only, not for human or veterinary use.

LUF5484 is an A1AR PAM

Chemical Structure

LUF5484
LUF5484
CAS#N/A

Theoretical Analysis

MedKoo Cat#: 125654

Name: LUF5484

CAS#: N/A

Chemical Formula: C15H13Cl2NOS

Exact Mass: 325.0100

Molecular Weight: 326.24

Elemental Analysis: C, 55.23; H, 4.02; Cl, 21.73; N, 4.29; O, 4.90; S, 9.83

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
LUF5484; LUF-5484; LUF 5484
IUPAC/Chemical Name
(2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)(3,4-dichlorophenyl)methanone
InChi Key
VBHZVGMOPSACQD-UHFFFAOYSA-N
InChi Code
InChI=1S/C15H13Cl2NOS/c16-10-6-5-8(7-11(10)17)14(19)13-9-3-1-2-4-12(9)20-15(13)18/h5-7H,1-4,18H2
SMILES Code
O=C(C1=C(N)SC2=C1CCCC2)C3=CC=C(Cl)C(Cl)=C3
Appearance
To be determined
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 326.24 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Bueters TJ, van Helden HP, Danhof M, IJzerman AP. Effects of the adenosine A1 receptor allosteric modulators PD 81,723 and LUF 5484 on the striatal acetylcholine release. Eur J Pharmacol. 2002 Nov 15;454(2-3):177-82. doi: 10.1016/s0014-2999(02)02494-9. PMID: 12421644. 2: Dalpiaz A, Pavan B, Ngos FN, Franchetti P, IJzerman AP. Temperature dependence of the affinity enhancement of selective adenosine A1 receptor agonism: a thermodynamic analysis. Eur J Pharmacol. 2002 Jul 19;448(2-3):123-31. doi: 10.1016/s0014-2999(02)01982-9. PMID: 12144931.