Synonym
RS23597-190 HCl; RS23597190 HCl; RS23597 190 HCl; RS23597-190 hydrochloride; RS23597190 hydrochloride; RS23597 190 hydrochloride;
IUPAC/Chemical Name
3-(piperidin-1-yl)propyl 4-amino-5-chloro-2-methoxybenzoate hydrochloride
InChi Key
QLZLBYYNMGQIAR-UHFFFAOYSA-N
InChi Code
InChI=1S/C16H23ClN2O3.ClH/c1-21-15-11-14(18)13(17)10-12(15)16(20)22-9-5-8-19-6-3-2-4-7-19;/h10-11H,2-9,18H2,1H3;1H
SMILES Code
O=C(OCCCN1CCCCC1)C2=CC(Cl)=C(N)C=C2OC.[H]Cl
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
|
Solvent |
mg/mL |
mM |
| Solubility |
| Water |
36.3 |
100.00 |
Note: There can be variations in solubility for the same chemical from different vendors or different batches from the same vendor. The following factors can affect the solubility of the same chemical: solvent used for crystallization, residual solvent content, polymorphism, salt versus free form, degree of hydration, solvent temperature. Please use the solubility data as a reference only. Warming and sonication will facilitate dissolving. Still have questions? Please contact our Technical Support scientists.
Preparing Stock Solutions
The following data is based on the
product
molecular weight
363.28
Batch specific molecular weights may vary
from batch to batch
due to the degree of hydration, which will
affect the solvent
volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass |
1 mg |
5 mg |
10 mg |
| 1 mM |
1.15 mL |
5.76 mL |
11.51 mL |
| 5 mM |
0.23 mL |
1.15 mL |
2.3 mL |
| 10 mM |
0.12 mL |
0.58 mL |
1.15 mL |
| 50 mM |
0.02 mL |
0.12 mL |
0.23 mL |
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6: Abe K, Fujimoto T, Akaishi T, Misawa M. Stimulation of basolateral amygdaloid serotonin 5-HT(2C) receptors promotes the induction of long-term potentiation in the dentate gyrus of anesthetized rats. Neurosci Lett. 2009 Feb 13;451(1):65-8. doi: 10.1016/j.neulet.2008.12.023. Epub 2008 Dec 24. PMID: 19110035.
7: Bonsi P, Cuomo D, Ding J, Sciamanna G, Ulrich S, Tscherter A, Bernardi G, Surmeier DJ, Pisani A. Endogenous serotonin excites striatal cholinergic interneurons via the activation of 5-HT 2C, 5-HT6, and 5-HT7 serotonin receptors: implications for extrapyramidal side effects of serotonin reuptake inhibitors. Neuropsychopharmacology. 2007 Aug;32(8):1840-54. doi: 10.1038/sj.npp.1301294. Epub 2007 Jan 3. PMID: 17203014.
8: Cao C, Han JH, Kim SZ, Cho KW, Kim SH. Diverse regulation of atrial natriuretic peptide secretion by serotonin receptor subtypes. Cardiovasc Res. 2003 Aug 1;59(2):360-8. doi: 10.1016/s0008-6363(03)00394-8. PMID: 12909319.
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