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MedKoo Cat#: 577325 | Name: Methoxyphenamine hydrochloride

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Methoxyphenamine hydrochloride inhibits basal and histamine-induced nasal congestion in anesthetized rats.

Chemical Structure

Methoxyphenamine hydrochloride
Methoxyphenamine hydrochloride
CAS#5588-10-3

Theoretical Analysis

MedKoo Cat#: 577325

Name: Methoxyphenamine hydrochloride

CAS#: 5588-10-3

Chemical Formula: C11H18ClNO

Exact Mass: 215.1077

Molecular Weight: 215.72

Elemental Analysis: C, 61.25; H, 8.41; Cl, 16.43; N, 6.49; O, 7.42

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Methoxiphenadrin hydrochloride; Methoxyphenamine hydrochloride; Methoxyphenamine HCl; Orthoxine hydrochloride
IUPAC/Chemical Name
Benzeneethanamine, 2-methoxy-N,alpha-dimethyl-, hydrochloride
InChi Key
FGSJNNQVSUVTPW-UHFFFAOYSA-N
InChi Code
InChI=1S/C11H17NO.ClH/c1-9(12-2)8-10-6-4-5-7-11(10)13-3;/h4-7,9,12H,8H2,1-3H3;1H
SMILES Code
Cl.CNC(C)Cc1ccccc1OC
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info
Toxicity Data: Dog - LD50, Subcutaneous (241 mg/kg) - Effects: None reported Mouse - LD50, Intraperitoneal (90 mg/kg) - Effect: None reported Mouse - LD50, Oral (605 mg/kg) - Effect: Dyspnea, Convulsions or effect on seizure threshold, Ataxia Mouse - LD50, Subcutaneous (380 mg/kg) - Effect: Dyspnea, Convulsions or effect on seizure threshold, Ataxia Rabbit - LD50, Intravenous (30 mg/kg) - No effects reported Rabbit - LD50, Oral (652 mg/kg) - No effects reported Rabbit - LD50, Subcutaneous (269 mg/kg) - No effects reported Rat - LD50, Intravenous (50 mg/kg) - No effects reported Rat - LD50, Oral (630 mg/kg) - No effects reported Rat - LD50, Subcutaneous (573 mg/kg) - No effects reported Sources: Nippon Yakurigaku Zasshi. Japanese Journal of Pharmacology. Vol. 54, Pg. 688, 1958. "Psychotropic Drugs and Related Compounds," 2nd ed., Usdin, E., and D.H. Efron, Washington, DC, 1972Vol. -, Pg. 348, 1972. Drugs in Japan Vol. 6, Pg. 837, 1982.

Preparing Stock Solutions

The following data is based on the product molecular weight 215.72 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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