OM-1700 is a novel potent and selective tankyrase inhibitor, showing a favorable ADME profile, including improved Caco-2 permeability and oral bioavailability in mice, and exhibiting antiproliferative efficacy in the colon cancer cell line COLO 320DM in vitro.
MedKoo Cat#: 464880
Name: OM-1700
CAS#: unknown
Chemical Formula: C25H23FN6O2
Exact Mass: 458.1867
Molecular Weight: 458.50
Elemental Analysis: C, 65.49; H, 5.06; F, 4.14; N, 18.33; O, 6.98
The following data is based on the product molecular weight 458.50 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
