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MedKoo Cat#: 575759 | Name: Tizanox

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tizanox is an anthelminthic.

Chemical Structure

Tizanox
CAS#147687-38-5

Theoretical Analysis

MedKoo Cat#: 575759

Name: Tizanox

CAS#: 147687-38-5

Chemical Formula: C18H24N2O3S

Exact Mass: 348.1508

Molecular Weight: 348.46

Elemental Analysis: C, 62.04; H, 6.94; N, 8.04; O, 13.77; S, 9.20

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
G-1587; G 1587; G1587; Tizanox
IUPAC/Chemical Name
(1,2,5)Thiadiazino(3,2-a)isoquinoline, 1,2,3,6,7,11b-hexahydro-2-(cyclohexylcarbonyl)-, 4,4-dioxide
InChi Key
YBCHDBKDRBCGTF-UHFFFAOYSA-N
InChi Code
InChI=1S/C18H24N2O3S/c21-18(15-7-2-1-3-8-15)19-12-17-16-9-5-4-6-14(16)10-11-20(17)24(22,23)13-19/h4-6,9,15,17H,1-3,7-8,10-13H2
SMILES Code
O=C(C1CCCCC1)N2CC3N(CCc4ccccc34)S(=O)(=O)C2
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 348.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1. Mikhaĭlitsyn FS, Sergovskaia NL, Uvarova NA, Lopatin BV, Gitsu GA, Astaf'ev BA, Lebedeva MN, Lychko ND. Tekhnologiia proizvodstva protivoparazitarnykh preparatov. 9. Novyĭ preparat tizanoks i otsenka ego protivogimenolepidoznoĭ aktivnosti [The technology for manufacturing antiparasitic preparations. 9. The new preparation tizanox and an evaluation of its anti-Hymenolepis activity]. Med Parazitol (Mosk). 1999 Jan-Mar;(1):49-51. Russian. PMID: 10414049. 2. Mikhaĭlitsyn FS, Kovalenko FP, Sergovskaia NL, Lebedeva MN, Dzhabarova VI, Lychko ND, Naĭdenova AS. Poisk novykh protivoparazitarnykh sredstv. 11. Ostraia toksichnost' i protivotsestodnaia aktivnost' novogo antigel'mintika tizanoksa v sravnenii s azinoksom [The search for new antiparasitic agents. 11. The acute toxicity and anticestodal activity of the new anthelmintic Tizanox compared with Azinox]. Med Parazitol (Mosk). 1992 Mar-Apr;(2):32-4. Russian. PMID: 1435534.