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MedKoo Cat#: 575713 | Name: Sepimostate mesilate

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Sepimostate mesilate is a biochemical used in therapy of pancreatitis.

Chemical Structure

Sepimostate mesilate
CAS#103926-82-5

Theoretical Analysis

MedKoo Cat#: 575713

Name: Sepimostate mesilate

CAS#: 103926-82-5

Chemical Formula: C23H27N5O8S2

Exact Mass: 565.1301

Molecular Weight: 565.62

Elemental Analysis: C, 48.84; H, 4.81; N, 12.38; O, 22.63; S, 11.34

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
FUT 187; FUT187; FUT-187; Sepimostate mesilate; Sepimostat mesylate; TO187; TO 187; TO-187
IUPAC/Chemical Name
Benzoic acid, 4-((4,5-dihydro-1H-imidazol-2-yl)amino)-, 6-(aminoiminomethyl)-2-naphthalenyl ester, dimethanesulfonate
InChi Key
NAMGRNXMZHEICS-UHFFFAOYSA-N
InChi Code
InChI=1S/C21H19N5O2.CH4O3S/c22-19(23)16-2-1-15-12-18(8-5-14(15)11-16)28-20(27)13-3-6-17(7-4-13)26-21-24-9-10-25-21;1-5(2,3)4/h1-8,11-12H,9-10H2,(H3,22,23)(H2,24,25,26);1H3,(H,2,3,4)
SMILES Code
CS(=O)(=O)O.NC(=N)c1ccc2cc(OC(=O)c3ccc(NC4=NCCN4)cc3)ccc2c1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 565.62 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1. Yuasa C, Irimura K, Oda M, Fukui K, Oka T. Oral administration of sepimostat mesilate prevents acute alcohol pancreatic injury in rats. J Pharm Pharmacol. 1999 Jul;51(7):867-71. doi: 10.1211/0022357991773087. PMID: 10467964. 2. Tsuruda A, Kanno S, Ohtani H, Suzuki R, Nishioka M, Koshiyama Y, Kurumi M. Effect of sepimostat mesilate on experimental venous thrombosis in rats. Thromb Res. 2001 Feb 1;101(3):193-201. doi: 10.1016/s0049-3848(00)00400-x. PMID: 11228342.