Cioteronel | CAS# 89672-11-7 | Anti-Androgen

MedKoo Cat#: 412926 | Name: Cioteronel

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Cioteronel is an antiandrogen agent which was in phase II trials for androgenetic alopecia.

Chemical Structure

Cioteronel

CAS#89672-11-7

Theoretical Analysis

MedKoo Cat#: 412926

Name: Cioteronel

CAS#: 89672-11-7

Chemical Formula: C16H28O2

Exact Mass: 252.2089

Molecular Weight: 252.39

Elemental Analysis: C, 76.14; H, 11.18; O, 12.68

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

Cioteronel; Cioteronelum; UNII-1RTH95874Z

IUPAC/Chemical Name

2(1H)-Pentalenone, hexahydro-4-(5-methoxyheptyl)-

InChi Key

KDULJHFMZBRAHO-UHFFFAOYSA-N

InChi Code

InChI=1S/C16H28O2/c1-3-15(18-2)7-5-4-6-12-8-9-13-10-14(17)11-16(12)13/h12-13,15-16H,3-11H2,1-2H3

SMILES Code

O=C1CC2CCC(CCCCC(OC)CC)C2C1

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 252.39 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Ford LC, Hammill HA, DeLange RJ, Bruckner DA, Suzuki-Chavez F, Mickus KL, Lebherz TB. Determination of estrogen and androgen receptors in Trichomonas vaginalis and the effects of antihormones. Am J Obstet Gynecol. 1987 May;156(5):1119-21. doi: 10.1016/0002-9378(87)90122-0. PMID: 3495180. 2: de Zeeuw RA, Herder RE, Wiechers JW, Drenth BF. Metabolic conversion of cyoctol during skin passage in humans. Pharm Res. 1990 Jun;7(6):638-43. doi: 10.1023/a:1015878430173. PMID: 2367332. 3: Ford LC, Kasha W, Chang NH, DeLange RJ. Antiandrogen and antineoplastic effects of a novel drug, CPC10997. Chemotherapy. 1985;31(5):362-5. doi: 10.1159/000238360. PMID: 3840430.