Cinuperone is an antagonist of D2, alpha1 adrenergic and sigma receptors. The drug selectively inhibits dopamine agonists-dependent behaviors, mediated by the limbic system. The clinical development of the drug as an antipsychotic was terminated due to orthostasis.
MedKoo Cat#: 412925
Name: Cinuperone
CAS#: 82117-51-9
Chemical Formula: C23H24FN3O
Exact Mass: 377.1903
Molecular Weight: 377.46
Elemental Analysis: C, 73.19; H, 6.41; F, 5.03; N, 11.13; O, 4.24
The following data is based on the product molecular weight 377.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
