BJG-03-025 is a Potent and Selective Focal Adhesion Kinase (FAK) Inhibitor BJG-03-025 displays potent biochemical FAK inhibition (IC50 = 20 nM), excellent kinome selectivity, activity in 3D-culture breast and gastric cancer models, and favorable pharmacokinetic properties in mice. BJG-03-025 is a valuable chemical probe for evaluation of FAK-dependent biology.
MedKoo Cat#: 463639
Name: BJG-03-025
CAS#: unknown
Chemical Formula: C28H37N9O2S
Exact Mass: 563.2791
Molecular Weight: 563.73
Elemental Analysis: C, 59.66; H, 6.62; N, 22.36; O, 5.68; S, 5.69
The following data is based on the product molecular weight 563.73 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
