MedKoo Cat#: 575304 | Name: Famiraprinium

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Famiraprinium is a competitive antagonist at the GABA receptor site.

Chemical Structure

Famiraprinium
Famiraprinium
CAS#105538-42-9

Theoretical Analysis

MedKoo Cat#: 575304

Name: Famiraprinium

CAS#: 105538-42-9

Chemical Formula: C15H17N3O2

Exact Mass: 271.1321

Molecular Weight: 271.32

Elemental Analysis: C, 66.40; H, 6.32; N, 15.49; O, 11.79

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
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Synonym
Famiraprinium
IUPAC/Chemical Name
4-(6-imino-5-methyl-3-phenylpyridazin-1(6H)-yl)butanoic acid
InChi Key
LLZVAIDABZBAGE-UHFFFAOYSA-N
InChi Code
InChI=1S/C15H17N3O2/c1-11-10-13(12-6-3-2-4-7-12)17-18(15(11)16)9-5-8-14(19)20/h2-4,6-7,10,16H,5,8-9H2,1H3,(H,19,20)
SMILES Code
CC1=CC(=NN(CCCC(=O)O)C1=N)c2ccccc2
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 271.32 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1. Worms P, Chambon JP, Biziere K. Behavioural evidence for a selective GABA-A antagonistic activity of SR 95103 and SR 42641 after intrastriatal injection in mice. Eur J Pharmacol. 1987 Jun 26;138(3):343-50. doi: 10.1016/0014-2999(87)90472-9. PMID: 3040438. 2. Santucci V, Fournier M, Chambon JP, Biziere K. Electroencephalographic study of SR 95103, a GABAA antagonist: interaction with inhibitory amino acids and muscimol. Eur J Pharmacol. 1985 Aug 15;114(2):219-22. doi: 10.1016/0014-2999(85)90630-2. PMID: 2995080. 3. Schmitt P, Di Scala G, Brandao ML, Karli P. Behavioral effects of microinjections of SR 95103, a new GABA-A antagonist, into the medial hypothalamus or the mesencephalic central gray. Eur J Pharmacol. 1985 Nov 5;117(2):149-58. doi: 10.1016/0014-2999(85)90599-0. PMID: 3000802.