NR162 is a novel potent and selective CASK inhibitor with a Kd of 22 nM in ITC and IC50 of 80 nM in NanoBRET assay.
MedKoo Cat#: 463265
Name: NR162
CAS#: 2755241-73-5
Chemical Formula: C23H28Br2N6O3
Exact Mass: 594.0590
Molecular Weight: 596.32
Elemental Analysis: C, 46.33; H, 4.73; Br, 26.80; N, 14.09; O, 8.05
The following data is based on the product molecular weight 596.32 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
