Synonym
Caf 603; Caf603; Caf-603
IUPAC/Chemical Name
1,2-Azulenediol, 1,2,3,3a,4,7,8,8a-octahydro-3a,6-dimethyl-1-(1-methylethyl)-, (1alpha,2alpha,3aalpha,8abeta)-(-)-
InChi Key
WBVHJGBFCZGJRZ-CBBWQLFWSA-N
InChi Code
InChI=1S/C15H26O2/c1-10(2)15(17)12-6-5-11(3)7-8-14(12,4)9-13(15)16/h7,10,12-13,16-17H,5-6,8-9H2,1-4H3/t12-,13+,14+,15-/m1/s1
SMILES Code
O[C@@]1(C(C)C)[C@@H](O)C[C@]2(C)CC=C(C)CC[C@@]12[H]
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
Preparing Stock Solutions
The following data is based on the
product
molecular weight
238.37
Batch specific molecular weights may vary
from batch to batch
due to the degree of hydration, which will
affect the solvent
volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass |
1 mg |
5 mg |
10 mg |
| 1 mM |
1.15 mL |
5.76 mL |
11.51 mL |
| 5 mM |
0.23 mL |
1.15 mL |
2.3 mL |
| 10 mM |
0.12 mL |
0.58 mL |
1.15 mL |
| 50 mM |
0.02 mL |
0.12 mL |
0.23 mL |
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2: Shi ZZ, Fang ST, Miao FP, Yin XL, Ji NY. Trichocarotins A-H and trichocadinin A, nine sesquiterpenes from the marine-alga-epiphytic fungus Trichoderma virens. Bioorg Chem. 2018 Dec;81:319-325. doi: 10.1016/j.bioorg.2018.08.027. Epub 2018 Aug 27. PMID: 30176571.
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5: Lee SH, Hensens OD, Helms GL, Liesch JM, Zink DL, Giacobbe RA, Bills GF, Stevens-Miles S, Garcia ML, Schmalhofer WA, et al. L-735,334, a novel sesquiterpenoid potassium channel-agonist from Trichoderma virens. J Nat Prod. 1995 Dec;58(12):1822-8. doi: 10.1021/np50126a004. PMID: 8691204.
6: Watanabe N, Yamagishi M, Mizutani T, Kondoh H, Omura S, Hanada K, Kushida K. CAF-603: a new antifungal carotane sesquiterpene. Isolation and structure elucidation. J Nat Prod. 1990 Sep-Oct;53(5):1176-81. doi: 10.1021/np50071a006. PMID: 2292685.
