BVT-74316 | CAS#917095-86-4 | antagonist of the serotonin 6 receptor (5-HT6)

MedKoo Cat#: 412163 | Name: BVT-74316

Description:

WARNING: This product is for research use only, not for human or veterinary use.

BVT-74316 is an orally administered antagonist of the serotonin 6 receptor (5-HT6) being developed by Proximagen

Chemical Structure

BVT-74316

CAS#917095-86-4

Theoretical Analysis

MedKoo Cat#: 412163

Name: BVT-74316

CAS#: 917095-86-4

Chemical Formula: C21H24N2O5S

Exact Mass: 416.1406

Molecular Weight: 416.49

Elemental Analysis: C, 60.56; H, 5.81; N, 6.73; O, 19.21; S, 7.70

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

BVT-74316; BVT74316; BVT 74316

IUPAC/Chemical Name

5-Benzofuransulfonamide, N-(2-methoxy-5-methylphenyl)-7-(4-piperidinyloxy)-

InChi Key

UPQJYTNALAIZCC-UHFFFAOYSA-N

InChi Code

InChI=1S/C21H24N2O5S/c1-14-3-4-19(26-2)18(11-14)23-29(24,25)17-12-15-7-10-27-21(15)20(13-17)28-16-5-8-22-9-6-16/h3-4,7,10-13,16,22-23H,5-6,8-9H2,1-2H3

SMILES Code

O=S(C1=CC(OC2CCNCC2)=C(OC=C3)C3=C1)(NC4=CC(C)=CC=C4OC)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 416.49 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Halford JC, Harrold JA, Boyland EJ, Lawton CL, Blundell JE. Serotonergic drugs : effects on appetite expression and use for the treatment of obesity. Drugs. 2007;67(1):27-55. doi: 10.2165/00003495-200767010-00004. PMID: 17209663.