GSK046, also known as iBET-BD2, is a highly selective inhibitor of the second bromodomains of the BET proteins that has undergone extensive pre-clinical in vitro and in vivo characterization.
MedKoo Cat#: 462853
Name: GSK046
CAS#: 2474876-09-8
Chemical Formula: C23H27FN2O4
Exact Mass: 414.1955
Molecular Weight: 414.48
Elemental Analysis: C, 66.65; H, 6.57; F, 4.58; N, 6.76; O, 15.44
The following data is based on the product molecular weight 414.48 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
