MedKoo Cat#: 534941 | Name: Tribendimidine
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tribendimidine (TBD) is a broad-spectrum anthelmintic drug that is also significantly effective in treating clonorchiasis. It is a derivative of amidantel. Tribendimidine was as effective as praziquantel against O. felineus liver flukes.

Chemical Structure

Tribendimidine
Tribendimidine
CAS#115103-15-6

Theoretical Analysis

MedKoo Cat#: 534941

Name: Tribendimidine

CAS#: 115103-15-6

Chemical Formula: C28H32N6

Exact Mass: 452.2688

Molecular Weight: 452.61

Elemental Analysis: C, 74.30; H, 7.13; N, 18.57

Price and Availability

Size Price Availability Quantity
25mg USD 450.00 2 Weeks
50mg USD 750.00 2 Weeks
100mg USD 1,250.00 2 Weeks
200mg USD 2,250.00 2 Weeks
500mg USD 3,650.00 2 Weeks
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Related CAS #
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Synonym
Tribendimidine
IUPAC/Chemical Name
Ethanimidamide, N',N'''-(1,4-phenylenebis(methylidynenitrilo-4,1-phenylene))bis(N,N-dimethyl-Tribendimidine
InChi Key
XOIOGKHKNQYULW-HTNNXBMUSA-N
InChi Code
InChI=1S/C28H32N6/c1-21(33(3)4)31-27-15-11-25(12-16-27)29-19-23-7-9-24(10-8-23)20-30-26-13-17-28(18-14-26)32-22(2)34(5)6/h7-20H,1-6H3/b29-19+,30-20+,31-21+,32-22+
SMILES Code
C/C(N(C)C)=N\C1=CC=C(/N=C/C2=CC=C(/C=N/C3=CC=C(/N=C(N(C)C)\C)C=C3)C=C2)C=C1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 452.61 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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PMID: 20118558. 11: Inoue A, Tamagawa-Mineoka R, Katoh N, Kishimoto S. Allergic contact dermatitis caused by tribenoside. Contact Dermatitis. 2009 Jun;60(6):349-50. doi: 10.1111/j.1600-0536.2009.01544.x. PMID: 19489977. 12: Aliev SA, Ibishov KG, Aliev ES. [Certain aspects of pathogenesis of hemorheological and trophic disturbances and their pharmacological correction in patients with chronic venous insufficiency]. Vestn Khir Im I I Grek. 2008;167(2):39-43. Russian. PMID: 18522184. 13: Hashizume H, Takigawa M. Drug-induced hypersensitivity syndrome associated with cytomegalovirus reactivation: immunological characterization of pathogenic T cells. Acta Derm Venereol. 2005;85(1):47-50. doi: 10.1080/00015550410024094. PMID: 15848991. 14: Endo H, Kawada A, Yudate T, Aragane Y, Yamada H, Tezuka T. Drug eruption due to tribenoside. Contact Dermatitis. 1999 Oct;41(4):223. doi: 10.1111/j.1600-0536.1999.tb06137.x. PMID: 10515105. 15: Chayen J, Bitensky L, Chambers MG. 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