MedKoo Cat#: 574424 | Name: TC-G 1000
Featured

Description:

WARNING: This product is for research use only, not for human or veterinary use.

TC-G 1000 is a selective α2D-adrenoceptor agonist that exhibits analgesic activity in a mouse model of abdominal irritation. It is orally active.

Chemical Structure

TC-G 1000
TC-G 1000
CAS#245744-18-7

Theoretical Analysis

MedKoo Cat#: 574424

Name: TC-G 1000

CAS#: 245744-18-7

Chemical Formula: C17H18N2O4S

Exact Mass: 346.0987

Molecular Weight: 346.40

Elemental Analysis: C, 58.95; H, 5.24; N, 8.09; O, 18.47; S, 9.26

Price and Availability

Size Price Availability Quantity
10mg USD 450.00 2 Weeks
50mg USD 1,150.00 2 Weeks
Bulk Inquiry
Buy Now
Add to Cart
Related CAS #
No Data
Synonym
TC-G 1000
IUPAC/Chemical Name
4-(6,7-Dihydro-1,3-dimethylbenzo[c]thien-4-yl)-1H-imidazole maleate
InChi Key
OPCJPAYHMCWCGW-BTJKTKAUSA-N
InChi Code
InChI=1S/C13H14N2S.C4H4O4/c1-8-10-4-3-5-11(12-6-14-7-15-12)13(10)9(2)16-8;5-3(6)1-2-4(7)8/h5-7H,3-4H2,1-2H3,(H,14,15);1-2H,(H,5,6)(H,7,8)/b;2-1-
SMILES Code
CC1=C2C(C(C3=CNC=N3)=CCC2)=C(C)S1.O=C(\C=C/C(O)=O)O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 346.40 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Ross et al (2000) α2 adrenoceptor agonists as potential analgesic agents. 2. Discovery of 4-(4-Imidazo)-1,3-dimethyl-6,7-dihydrothianaphthene as a high-affinity ligand for the α2D adrenergic receptor. J.Med.Chem. 43 1423 PMID: 10715142 Gordon, A. N., Teneriello, M. G., Spirtos, N., Janicek, M. F., Goss, T., Wang, Y., ... & Tai, D. F. (2008). Phase III trial of induction gemcitabine (G) or paclitaxel (T) plus carboplatin (C) followed by elective T consolidation in advanced ovarian cancer (OC): Interim analysis of induction chemotherapy. Journal of Clinical Oncology, 26(15_suppl), 5536-5536.