CAY10762 | CAS#2514-37-6 | monoacylglycerol lipase inhibitor

MedKoo Cat#: 462148 | Name: CAY10762

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Description:

WARNING: This product is for research use only, not for human or veterinary use.

CAY10762 is an inhibitor of monoacylglycerol lipase. It reduces hydrogen peroxide-induced lactate dehydrogenase (LDH) release from Neuro2a cells when used at a concentration of 1 µM.

Chemical Structure

CAY10762

CAS#2514-37-6

Theoretical Analysis

MedKoo Cat#: 462148

Name: CAY10762

CAS#: 2514-37-6

Chemical Formula: C15H13NOS

Exact Mass: 255.0718

Molecular Weight: 255.34

Elemental Analysis: C, 70.56; H, 5.13; N, 5.49; O, 6.27; S, 12.56

Price and Availability

Size	Price	Availability	Quantity
5mg	USD 425.00	2 Weeks
10mg	USD 765.00	2 Weeks

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Related CAS #

No Data

Synonym

CAY10762; CAY 10762; CAY-10762

IUPAC/Chemical Name

2-phenethylbenzo[d]isothiazol-3(2H)-one

InChi Key

VUMUTUGUKRGYGW-UHFFFAOYSA-N

InChi Code

InChI=1S/C15H13NOS/c17-15-13-8-4-5-9-14(13)18-16(15)11-10-12-6-2-1-3-7-12/h1-9H,10-11H2

SMILES Code

O=C1C2=CC=CC=C2SN1CCC3=CC=CC=C3

Appearance

Solid powder

Purity

>95% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

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Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 255.34 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Castelli, R., Scalvini, L., Vacondio, F., et al. Benzisothiazolinone derivatives as potent allosteric monoacylglycerol lipase inhibitors that functionally mimic sulfenylation of regulatory cysteines. J. Med. Chem. 63(3), 1261-1280 (2020).