9-Me-1 is a novel, potent, mutant-selective BET bromodomain inhibitor, showing >100-fold selectivity for the L/V mutant over wild-type and excellent DMPK properties.
MedKoo Cat#: 533782
Name: 9-Me-1
CAS#: N/A
Chemical Formula: C22H21ClN4O3
Exact Mass: 424.1302
Molecular Weight: 424.89
Elemental Analysis: C, 62.19; H, 4.98; Cl, 8.34; N, 13.19; O, 11.30
The following data is based on the product molecular weight 424.89 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
