MedKoo Cat#: 585092 | Name: Tameridone

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tameridone is a sedative used for cattle.

Chemical Structure

Tameridone
Tameridone
CAS#102144-78-5

Theoretical Analysis

MedKoo Cat#: 585092

Name: Tameridone

CAS#: 102144-78-5

Chemical Formula: C22H26N6O2

Exact Mass: 406.2117

Molecular Weight: 406.49

Elemental Analysis: C, 65.01; H, 6.45; N, 20.68; O, 7.87

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Tameridone; R 51163; R 51 163
IUPAC/Chemical Name
1H-Purine-2,6-dione, 3,7-dihydro-7-(2-(4-(1H-indol-3-yl)-1-piperidinyl)ethyl)-1,3-dimethyl-
InChi Key
OJOSYHJYEWUYGU-UHFFFAOYSA-N
InChi Code
InChI=1S/C22H26N6O2/c1-25-20-19(21(29)26(2)22(25)30)28(14-24-20)12-11-27-9-7-15(8-10-27)17-13-23-18-6-4-3-5-16(17)18/h3-6,13-15,23H,7-12H2,1-2H3
SMILES Code
O=C(N1C)N(C)C2=C(N(CCN3CCC(C4=CNC5=C4C=CC=C5)CC3)C=N2)C1=O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 406.49 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Haigh JC, Gates CC. Capture of wood bison (Bison bison athabascae) using carfentanil-based mixtures. J Wildl Dis. 1995 Jan;31(1):37-42. PubMed PMID: 7563422. 2: Renecker LA, Bertwistle J, Kozak HM, Hudson RJ, Chabot D, MacLean S. R51163 as a sedative for handling and transporting plains bison and wapiti. J Wildl Dis. 1992 Apr;28(2):236-41. PubMed PMID: 1602574. 3: Schwartz CC, Hundertmark KJ, Lance WR. Effects of R51163 on intake and metabolism in moose. J Wildl Dis. 1991 Jan;27(1):119-22. PubMed PMID: 2023310. 4: Jiang YQ, Zuo CX. [Studies of chemical constituents from Tamarix chinensis Lour]. Yao Xue Xue Bao. 1988;23(10):749-55. Chinese. PubMed PMID: 3257027. 5: Degryse AD, Ooms LA. Clinical evaluation of R 51163, a new sedative in cattle. J Vet Pharmacol Ther. 1986 Dec;9(4):376-84. PubMed PMID: 3806779.