MedKoo Biosciences, Inc.
Tel:   +1-919-636-5577    Fax:   +1-919-980-4831    Email:   sales@medkoo.com
Search
Login Register
Search
MedKoo Cat#: 558701 | Name: FAUC150

Description:

WARNING: This product is for research use only, not for human or veterinary use.

FAUC150 is an irreversible dopamine D2 receptor ligand which covalently binds the L94C mutant of the dopamine D2 receptor.

Chemical Structure

FAUC150
FAUC150
CAS#NONE

Theoretical Analysis

MedKoo Cat#: 558701

Name: FAUC150

CAS#: NONE

Chemical Formula: C22H32N2O4S2

Exact Mass: 452.1803

Molecular Weight: 452.63

Elemental Analysis: C, 58.38; H, 7.13; N, 6.19; O, 14.14; S, 14.17

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
No Data
Synonym
FAUC-150; FAUC 150; FAUC150
IUPAC/Chemical Name
4-(2-((4-(3-((2-Aminoethyl)disulfaneyl)propoxy)-3-methoxyphenethyl)amino)ethyl)benzene-1,2-diol
InChi Key
VOOGOCKGMWMTJZ-UHFFFAOYSA-N
InChi Code
InChI=1S/C22H32N2O4S2/c1-27-22-16-18(4-6-21(22)28-12-2-13-29-30-14-9-23)8-11-24-10-7-17-3-5-19(25)20(26)15-17/h3-6,15-16,24-26H,2,7-14,23H2,1H3
SMILES Code
OC1=CC=C(CCNCCC2=CC=C(OCCCSSCCN)C(OC)=C2)C=C1O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 452.63 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Schwalbe T, Kaindl J, Hübner H, Gmeiner P. Potent haloperidol derivatives covalently binding to the dopamine D2 receptor. Bioorg Med Chem. 2017 Oct 1;25(19):5084-5094. doi: 10.1016/j.bmc.2017.06.034. Epub 2017 Jun 20. PubMed PMID: 28666858.