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MedKoo Cat#: 573283 | Name: Thenalidine

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Thenalidine is an antihistamine and antipruritic.

Chemical Structure

Thenalidine
Thenalidine
CAS#86-12-4

Theoretical Analysis

MedKoo Cat#: 573283

Name: Thenalidine

CAS#: 86-12-4

Chemical Formula: C17H22N2S

Exact Mass: 286.1504

Molecular Weight: 286.44

Elemental Analysis: C, 71.29; H, 7.74; N, 9.78; S, 11.19

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
AS 716, Sanbosten, Thenalidine, Thenophenopiperidine
IUPAC/Chemical Name
1-Methyl-4-N-2-thenylanilinopiperidine
InChi Key
KLOHYVOVXOUKQI-UHFFFAOYSA-N
InChi Code
1S/C17H22N2S/c1-18-11-9-16(10-12-18)19(14-17-8-5-13-20-17)15-6-3-2-4-7-15/h2-8,13,16H,9-12,14H2,1H3
SMILES Code
s1cccc1CN(c1ccccc1)C1CCN(C)CC1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 286.44 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Kleinrok Z, Jagiello-Wójtowicz E, Kolasa K. The central action of histamine. 3. The effect of antazoline and thenalidine on the brain noradrenaline and 5-hydroxytryptamine levels and behavior of rats receiving histamine intraventricularly. Pol J Pharmacol Pharm. 1973 Nov-Dec;25(6):519-24. PubMed PMID: 4151860. 2: GETZLER NA, EREAUX LP. Evaluation of thenalidine tratrate (sandostene) in dermatological disorders. Can Med Assoc J. 1959 Mar 15;80(6):445-8. PubMed PMID: 13629433; PubMed Central PMCID: PMC1830689. 3: ADAMS DA, PERRY S. Agranulocytosis associated with thenalidine (sandostene) tartrate therapy; report of three cases. J Am Med Assoc. 1958 Jul 5;167(10):1207-10. PubMed PMID: 13549246.