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MedKoo Cat#: 564671 | Name: HIF-1α-p300 PPI inhibitor-3

Description:

WARNING: This product is for research use only, not for human or veterinary use.

HIF-1α-p300 PPI inhibitor-3 is a small-molecule proteomimetic HIF-1alpha-p300 protein protein interaction inhibitor.

Chemical Structure

HIF-1α-p300 PPI inhibitor-3
HIF-1α-p300 PPI inhibitor-3
CAS#NONE

Theoretical Analysis

MedKoo Cat#: 564671

Name: HIF-1α-p300 PPI inhibitor-3

CAS#: NONE

Chemical Formula: C32H39N3O7

Exact Mass: 577.2788

Molecular Weight: 577.68

Elemental Analysis: C, 66.53; H, 6.81; N, 7.27; O, 19.39

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
HIF 1α p300 PPI inhibitor 3; HIF1αp300 PPI inhibitor-3; HIF-1α-p300 PPI inhibitor-3
IUPAC/Chemical Name
4-[4-(4-Amino-3-tert-butoxy-benzoylamino)-3-tert-butoxy-benzoylamino]-3-isopropoxy-benzoic acid
InChi Key
WNOWHWZFCTYSBC-UHFFFAOYSA-N
InChi Code
InChI=1S/C32H39N3O7/c1-18(2)40-26-17-21(30(38)39)11-14-23(26)34-29(37)20-10-13-24(27(16-20)42-32(6,7)8)35-28(36)19-9-12-22(33)25(15-19)41-31(3,4)5/h9-18H,33H2,1-8H3,(H,34,37)(H,35,36)(H,38,39)
SMILES Code
O=C(O)C1=CC=C(NC(C2=CC=C(NC(C3=CC=C(N)C(OC(C)(C)C)=C3)=O)C(OC(C)(C)C)=C2)=O)C(OC(C)C)=C1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 577.68 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Burslem GM, Kyle HF, Breeze AL, Edwards TA, Nelson A, Warriner SL, Wilson AJ. Small-molecule proteomimetic inhibitors of the HIF-1α-p300 protein-protein interaction. Chembiochem. 2014 May 26;15(8):1083-7. doi: 10.1002/cbic.201400009. Epub 2014 Apr 29. PubMed PMID: 24782431; PubMed Central PMCID: PMC4159589.

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