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MedKoo Cat#: 564636 | Name: ASP6432
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

ASP6432 is a potent and selective Type 1 Lysophosphatidic Acid (LPA1) receptor antagonist.

Chemical Structure

ASP6432
ASP6432
CAS#1282549-08-9

Theoretical Analysis

MedKoo Cat#: 564636

Name: ASP6432

CAS#: 1282549-08-9

Chemical Formula: C25H29KN4O7S2

Exact Mass: 600.1115

Molecular Weight: 600.75

Elemental Analysis: C, 49.98; H, 4.87; K, 6.51; N, 9.33; O, 18.64; S, 10.67

Price and Availability

Size Price Availability Quantity
5mg USD 650.00 2 Weeks
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Related CAS #
No Data
Synonym
ASP-6432; ASP 6432; ASP6432
IUPAC/Chemical Name
potassium (N-ethylsulfamoyl)(2-((4-hydroxy-3,5-dimethoxy-N-(3-phenylpropyl)benzamido)methyl)-1l3,3l2-thiazole-4-carbonyl)amide
InChi Key
HJDUIXQAOQSISD-UHFFFAOYSA-M
InChi Code
InChI=1S/C25H30N4O7S2.K/c1-4-26-38(33,34)28-24(31)19-16-37-22(27-19)15-29(12-8-11-17-9-6-5-7-10-17)25(32)18-13-20(35-2)23(30)21(14-18)36-3;/h5-7,9-10,13-14,16,26H,4,8,11-12,15H2,1-3H3,(H2,28,30,31,32);/q;+1/p-1
SMILES Code
O=C(C1=CC(OC)=C(O)C(OC)=C1)N(CC2=[S]C=C(C(N(S(=O)(NCC)=O)[K])=O)[N]2)CCCC3=CC=CC=C3
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 600.75 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Sakamoto K, Noguchi Y, Ueshima K, Yamakuni H, Ohtake A, Sato S, Ishizu K, Hosogai N, Kawaminami E, Takeda M, Masuda N. Effect of ASP6432, a Novel Type 1 Lysophosphatidic Acid Receptor Antagonist, on Urethral Function and Prostate Cell Proliferation. J Pharmacol Exp Ther. 2018 Aug;366(2):390-396. doi: 10.1124/jpet.118.247908. Epub 2018 Jun 8. PubMed PMID: 29884626.